Physicochemical properties in relation to biological action, Unit-I B.Pharm 4th Semester Notes PDF
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11/30/2020 06:13:00 PM
- Introduction to Medicinal Chemistry
- History and development of medicinal chemistry
- Physicochemical properties in relation to biological action
- Ionization, Solubility, Partition Coefficient, Hydrogen bonding, Protein binding, Chelation, Bioisosterism, Optical and Geometrical isomerism.
- Drug metabolisam
- Drug metabolism principles- Phase I and Phase II.
- Factors affecting drug metabolism including stereo chemical aspects
Physicochemical properties in relation to biological action
- Ionization
- Solubility
- Partition Coefficient
- Hydrogen bonding
- Protein binding
- Chelation
- Bioisosterism
- Optical and Geometrical isomerism
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